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化合物成分:刺五加甙(eleutheroside)A、B、B1、C、D、E,刺五加甙A即是胡蘿卜甙(daucosterol),刺五加甙B即是丁香甙(syringin)、芥子醛葡萄糖甙(sinapaldehyde glucoside),松柏醛葡萄糖甙(coniferaldehyde glucoside),松柏甙(coniferin),鵝掌楸甙(liriodemdrin),苦杏仁甙(amygdalin),3β-[O-β-D-吡喃葡萄糖基(1→3)-O-β-D-吡喃半乳糖基(1→4)-[O-α-L-吡喃鼠李糖基-(1→2)]-O-β-D-吡喃葡萄糖醛酸基]-16α-羥基-13β,28-環(huán)氧齊墩果烷{3β-[O-β-D-glucopyranosyl-(1→3)-O-β-D-galactopyranosyl-(1→4)-[O-α-L-rhamnopyranosyl-(1→2)]-O-β-D-glucoronopyranosyl]-16α-hydroxy-13β,28-epoxyoleanane},3β-[O-α-L-吡喃鼠李糖基(1→4)-O-α-L-吡喃鼠李糖基(1→4)-[O-α-L-吡喃鼠李糖基-(1→2)]-β-D-吡喃葡萄糖基-(1→x)-O-β-D-吡喃葡萄糖醛酸基]-16α-羥基-13β,28-環(huán)氧齊墩果烷{3β-[O-α-L-rhamnopyranosyl-(1→4)-O-α-L-rhamnopyranosyl(1→4)[O-α-L-rhamnopyranosyl(1→2)]-O-β-D-glucopyranosyl(1→x)-O-β-D-glucoronopyranosyl]-16α-hydroxy-13β,28-epoxyoleanane},芝麻素(seasamin),松柏醛(coniferylaldehyde),香草醛(vanillin),異秦皮定(isofraxidin),丁香樹脂酚(syringaresinol),丁香酸(syringic acid),香草酸(vanillic acid),羥基苯甲酸(hydroxybenzoic acid),對-香豆酸(p-coumaric acid),阿魏酸(ferulic acid),綠原酸(chlorogenic acid),咖啡酸(caffeic acid),1,5-二-O-咖啡酰奎寧酸(1,5-di-O-caffeoylquinic acid),油酸甲酯(methyloleate),油酸乙酯(ethyloleate),10,13-十八碳二烯酸甲酯(10,13-octadecadienoic acid methylester),10,13-十八碳二烯酸乙酯(10,13-octadecadienoic acid ethyl ester),9,11-十八碳二烯酸(9,11-octadecadienoic acid),十六碳三烯酸(hexadecatrienoic acid),肉豆蔻酸(myristic acid),棕櫚酸(palmitic acid),硬脂酸(stearic acid),白樺脂酸(betulic acid)及β-谷甾醇(β-sitosterol),刺五加多糖AS-Ⅱ、AS-Ⅲ及水溶性刺五加多糖PES-A、PES-B,異秦皮定-7-O-β-D-葡萄糖甙(isofraxidin-7-O-β-D-glucoside)即刺五加甙B1,丁香甙,右旋-丁香樹脂酚-二-O-β-D葡萄糖甙(syringaresinol-di-O-β-D-glucoside),右旋-丁香樹脂酚-O-β-D-葡萄糖甙(syringaresinol-O-β-D-glucoside),右旋-松脂酚-二-O-β-D-葡萄糖甙(pinoresinol-di-O-β-D-glucoside),右旋-松脂酚-O-β-D-葡萄糖甙(pinoresinol-O-β-D-glucoside),右旋-杜仲松脂酚-二-O-β-D-葡萄糖甙(medioresinol-di-O-β-D-glucoside),異秦皮定、綠原酸及2,6-二甲氧基苯醌(2,6-dimethoxybenzoquinone),刺五加甙I、K、L、M,刺五加葉甙(ciwujianoside)A1、A2、A3、A4、B、C1、C2、C3、C4、D1、D2、D3、E,常春藤皮甙B(hederasaponin B)齊墩果酸-3-α-吡喃鼠李糖基(1→2)-O-α-吡喃阿拉伯糖甙[3-O-α-rhamnopyranosyl(1→2)-arabinopyranosyl oleanolic acid]及30-去甲-12,20(29)-齊墩果二烯-28-酸-3-O-α-吡喃阿拉伯糖甙[3-O-α-arabinopyranosyl-30-norolean-12,20(29)-dien-28-oic acid],金絲桃甙(hyperin),3,4-二羥基苯甲酸(3,4-dihydroxy benzoic acid)。
藥理作用:具較人參更好的適應原樣作用。能增強機體抵抗力,延遲腫瘤發(fā)生,阻止腫瘤轉移,降低自發(fā)性腫瘤的形成過程等;調節(jié)病理過程,使其趨向于正?;淖饔?。
★改善神經系統(tǒng)功能
★抗疲勞、耐缺氧
★抗腫瘤
★阻止免疫功能下降、調節(jié)內分泌功能紊亂
★抗炎、抗菌、抗病毒
★抑制血小板聚集
★止咳 |