
1995年?畢業(yè)于華東理工大學(xué)精細(xì)化工系;
1998年?中國科學(xué)院上海有機(jī)化學(xué)研究所獲碩士學(xué)位;
2003年?美國賓夕法尼亞州立大學(xué)獲博士學(xué)位;
2003-2005年?美國Scripps研究所從事博士后研究;
2005-2009年?美國Boehringer Ingelheim任高級科學(xué)家;
2009-2011年?美國Boehringer Ingelheim任首席科學(xué)家;
2011年-至今?中國科學(xué)院上海有機(jī)化學(xué)研究所研究員、課題組長;同時兼任上??萍即髮W(xué)物質(zhì)學(xué)院教授、博導(dǎo);杭州高等研究院首席教授;華東理工大學(xué)藥學(xué)院博導(dǎo)。
發(fā)展新型高效的不對稱催化反應(yīng);
對具有重要生理活性的復(fù)雜天然產(chǎn)物的全合成;
發(fā)展高效、經(jīng)濟(jì)、綠色的藥物新工藝。
2024年獲英國皇家化學(xué)會Organic Division Horizon Prize
2023年中國科學(xué)院朱李月華優(yōu)秀教師獎
2019年入選國家相關(guān)人才計劃
2019年藥明康德生命化學(xué)研究獎學(xué)者
2018年科技部中青年科技創(chuàng)新領(lǐng)軍人才
2017年獲國家杰出青年基金資助
2015年獲第三屆全國均相催化青年獎
2013年入選上?!捌纸瞬拧庇媱?/span>
2012年獲Thieme Journal Award
2009年獲美國Boehringer Ingelheim 藥業(yè)公司President’s Award for Individual Excellence
1.?“Chiral Polymeric Diamine Ligands for Iridium-Catalyzed Asymmetric Transfer Hydrogenation” Yaodong Lin, Guangqing Xu* Wenjun Tang*. J. Am. Chem. Soc.?2024, 146, 27736-27744.
2.?“Rhodium-Catalyzed Asymmetric Reductive Hydroformylation of α-Substituted Enamides” Yuxin Zhu,§ Yuchen Zhang,§ Dongyang He, He Yang,* Xiao-Song Xue,* Wenjun Tang*. J. Am. Chem. Soc.?2024, 146, 33249-33257.
3.?“Dienediamine: A Safe Herbicide as Paraquat Surrogate” Henian Peng,§ Dake Zhao,§ Wenjun Tang,*Ai Peng* Mol. Plant.?2023, 16, 1962-1975.
4.?“Enantioselective transformations in the synthesis of therapeutic agents” He Yang,§ Hanxiao Yu,§ Izabela A. Stolarzewicz,* Wenjun Tang*?Chem. Rev.?2023, 123, 9397-9446.
5.?“Asymmetric Synthesis of Vicinal Tetrasubstituted Diamines via Reductive Coupling of Ketimines Templated by Chiral Diborons” Mingkang Zhou,§ Yaodong Lin,§ Xiao-Xuan Chen,§ Guangqing Xu,* Lung Wa Chung,* Wenjun Tang*?Angew. Chem., Int. Ed.?2023, 62, e202300334.
6.?“Heck Reaction of N-Heteroaryl Halides for Concise Synthesis of Chiral α-Heteroaryl-substituted Heterocycles” Bowen Li, Bangke Luo, He Yang,* Wenjun Tang* Angew. Chem., Int. Ed.?2022, 61, e202209087.
7.?“Enantioselective Construction of ortho-Sulfur- or Nitrogen-Substituted Axially Chiral Biaryls and Asymmetric Synthesis of Isoplagiochin D” He Yang, Wenjun Tang* Nat. Commun.?2022, 13, 4577.
8.?“Enantioselective α-Carbonylative Arylation for Facile Construction of Chiral Spirocyclic β,β'‐Diketones” Ting Wu, Qinghai Zhou, Wenjun Tang* Angew. Chem., Int. Ed.?2021, 60, 9978-9983.
9.?“Asymmetric Hydroesterification of Diarylmethyl Carbinols” Duanshuai Tian, Ronghua Xu, Jinbin Zhu, Jianxun Huang, Wei Dong, Jerome Claverie, Wenjun Tang* Angew. Chem., Int. Ed. 2021, 60, 6305-6309.
10.?“Enantioselective Reductive Coupling of Imines Templated by Chiral Diboron” Mingkang Zhou, Kaidi Li, Dongping Chen, Ronghua Xu, Guangqing Xu, *Wenjun Tang* J. Am. Chem. Soc.?2020, 142, 10337-10342.
11.?“Enantioselective Cross-Coupling for Axially Chiral Tetra-ortho-Substituted Biaryls and Asymmetric Synthesis of Gossypol” He Yang, Jiawei Sun,?Wei Gu, Wenjun Tang* J. Am. Chem. Soc.?2020, 142, 8036–8043.
12.?“Expedite Construction of Various Bridged Polycyclic Skeletons by Palladium-Catalyzed Dearomatization” Xingye Mu, Hanxiao Yu, Henian Peng, Wenrui Xiong, Ting Wu, Wenjun Tang* Angew. Chem., Int. Ed.?2020, 59, 8143-8147.
13.?“Enantioselective Rhodium-Catalyzed Addition of Arylboroxines to N-Unprotected Ketimines: Efficient Synthesis of Cipargamin” Jinbin Zhu, Linwei Huang, Wei Dong, Naikai Li, Xingxin Yu, Wei-Ping Deng, Wenjun Tang* Angew. Chem., Int. Ed.?2019, 58, 16119-16123.
14.?“Stereoelectronic Effects in Ligand Design: Enantioselective RhodiumCatalyzed Hydrogenation of Aliphatic Cyclic Tetrasubstituted Enamides and Concise Synthesis of (R)-Tofacitinib” Chengxi Li,§?Feng Wan,§?Yuan Chen, Henian Peng, Wenjun Tang,* Shu Yu,* J. Christopher McWilliams,* Jason Mustakis, Lacey Samp, Robert J. Maguire, Angew. Chem., Int. Ed.?2019, 58, 13573-13583.
15.?“Enantioselective Palladium-Catalyzed Cross-Coupling of α-Bromo Carboxamides and Aryl Boronic Acids” Bowen Li, Tiejun Li, Muinat A. Aliyu, Zhen Hua Li, Wenjun Tang* Angew. Chem., Int. Ed. 2019, 58, 11355-11359.
16.?“Efficient Synthesis of (-)-Corynoline by Enantioselective Palladium Catalyzed α-Arylation with Sterically Hindered Substrates” Xiaofeng Rao,§ Naikai, Li,§ Heng Bai,§ Chaodi Dai, Zheng Wang, Wenjun Tang* Angew. Chem. Int. Ed.?2018, 57, 12328-12332.
17.?“Stereospecific Nucleophilic Substitution with Arylboronic Acids as Nucleophiles in the Presence of a CONH Group” Duanshuai Tian,§ Chengxi Li,§ Guoxian Gu, Henian Peng, Xumu Zhang,* Wenjun Tang* Angew. Chem. Int. Ed. 2018, 57, 7176-7180.
18.?“Practical and Asymmetric Reductive Coupling of Isoquinolines Templated by Chiral Diborons” Dongping Chen, Guangqing Xu, Qinghai Zhou, Lung Wa Chung, Wenjun Tang* J. Am. Chem. Soc.?2017, 139, 9767-9770.
19.?“Efficient Enantioselective Syntheses of (+)-Dalesconol A & B” Guoqing Zhao, § Guangqing Xu, § Chao Qian, Wenjun Tang* J. Am. Chem. Soc.?2017, 139,?3360-3363.
20.?Transition-Metal-Free Stereospecific Cross-Coupling with Alkenylboronic Acids as Nucleophiles” Chengxi Li, Yuanyuan Zhang, Qi Sun, Tongnian Gu, Henian Peng, Wenjun Tang* J. Am. Chem. Soc. 2016, 138, 10774-10777.
21.?“Highly Enantioselective Rhodium-Catalyzed Addition of Arylboroxines to Simple Ketones: Efficient Synthesis of Escitalopram” Linwei Huang, Jinbin Zhu, Guangjun Jiao, Zheng Wang, Xinxin Yu, Wei-Ping Deng,* Wenjun Tang* Angew. Chem., Int. Ed. 2016, 55, 4527.
22.?“Synthesis of Chiral 1,4-Benzodioxanes and Chromans by Enantioselective Palladium-Catalyzed Alkene Aryloxyarylation” Naifu Hu, Ke Li, Zheng Wang, Wenjun Tang* Angew. Chem., Int. Ed. 2016, 55, 5044.
23.?“Synthesis of Chiral α-Amino Tertiary Boronic Esters by Enantioselective Hydroboration of α-Arylenamides” Naifu Hu,§ Guoqing Zhao,§ Yuanyuan Zhang, Xiangqian Liu, Guangyu Li, Wenjun Tang* J. Am. Chem. Soc.?2015, 137,?6746-6749.
24.?“Enantioselective Palladium-Catalyzed Dearomative Cyclization for Efficient Synthesis of Terpenes and Steroids” Kang Du, Pan Guo, Yuan Chen, Zheng Cao, Wenjun Tang* Angew. Chem., Int. Ed.?2015, 54, 3033.
25.?“Efficient Syntheses of Sterically Hindered Acyclic Secondary Alkyl Arenes by Suzuki-Miyaura Cross-Couplings” Chengxi Li, Tianyu Chen, Guolan, Xiao, Bowen Li, Wenjun Tang*?Angew. Chem., Int. Ed.?2015, 54, 3792.
26.?“Highly Enantioselective Nickel-Catalyzed Intramolecular Reductive Cyclization of Alkynone” Wenzhen Fu, Ming Nie, Aizhen Wang, Wenjun Tang* Angew. Chem., Int. Ed. 2015, 54, 2520.
1. 國家重點(diǎn)研發(fā)計劃課題:鈀催化偶聯(lián)及催化劑創(chuàng)制,2022年-2027年。
2. 國家自然科學(xué)基金科學(xué)中心項目:神經(jīng)系統(tǒng)疾病致病機(jī)理的研究和干預(yù),2022年-2026年。
3. 國家杰出青年科學(xué)基金:催化不對稱合成,2018年-2022年。
4. 國家重點(diǎn)研發(fā)計劃課題:高端金屬與配體研制及關(guān)鍵技術(shù)研發(fā),2021年-2025年。
5. 廣東省重點(diǎn)領(lǐng)域研發(fā)計劃項目:三聯(lián)芳膦鈀碳氮偶聯(lián)催化劑的研發(fā)及產(chǎn)業(yè)化,2020年-2024年。
6. 上海市科委國家合作項目:有關(guān)磺酸化手性膦配體的材料科學(xué),2018年-2020年。
7. 國家自然科學(xué)基金面上項目:新型膦配體的發(fā)展2012年-2015年。
8. 國家自然科學(xué)基金重點(diǎn)項目:新型、高效P-手性配體的基礎(chǔ)和應(yīng)用研究2015年-2019年。
9. 國家自然科學(xué)基金面上項目:不對稱環(huán)化反應(yīng)方法學(xué)以及在天然產(chǎn)物和藥物合成中的應(yīng)用,2016年-2019年。
10. 中國科學(xué)院戰(zhàn)略性先導(dǎo)科技專項(B類):結(jié)構(gòu)與功能導(dǎo)向的新物質(zhì)創(chuàng)制,2016年-2021年。
11.?中國科學(xué)院前沿科學(xué)重點(diǎn)研究項目:配體促進(jìn)的高效偶聯(lián)反應(yīng)研究,2016年-2021年。

