
2006.09-2010.06??華中科技大學 ??????????????????理學學士
2010.09-2015.06??中國科學院上海有機化學研究所???理學博士???????導師:林國強?
2015.07-2016.01??中國科學院上海有機化學研究所???助理研究員?????導師:林國強?
2016.01-2019.11??美國加州大學伯克利分校 ??????????博士后???????導師:John F. Hartwig
2019.12-至今??????中國科學院上海有機化學研究所???研究員、課題組長、博士生導師
1. 不對稱催化合成:非經典的不對稱??3-取代
2. 糖、核酸的合成和修飾
2025 ??中國科學院人才計劃終期評估優(yōu)秀
2024 ??上??萍枷到y(tǒng)五四青年獎章
2024???Organic Chemistry Frontiers Emerging Investigator
2022? ?Thieme Chemistry Journals Award
2020? ?上海市科技青年啟明星計劃
2020 ??國家海外高層次人才計劃
20.?Gao-Liang Zheng, Yuchen Zhang, Jing-Ming Zhang, Liang Chen, Xiao-Song Xue*, Zhi-Tao He*.?Stereogenic P(V) Synthesis via Catalytic Continuous Substitutions.?J. Am. Chem. Soc.?2025,?147,?13566–13576.
19.?Xuan Zhang, Xian-Xiao Chen, Zi-Han Li, Guo-Qiang Lin, Zhi-Tao He*. Stereoselective P(III)-Glycosylation for the Preparation of Phosphinated Sugars.?Angew. Chem. Int. Ed.?2025,?64, e202420355.
18.?Ming-Qiao Tang, Zi-Jiang Yang, Ai-Jun Han, Zhi-Tao He*.?Diastereoselective and Enantioselective Hydrophosphinylations of Conjugated Enynes, Allenes and Dienes?via Synergistic Pd/Co Catalysis.?Angew. Chem. Int. Ed.?2025,?64,?e202413428.
17.?Yuan-Xiang Yang,?Yi-Fan Wang,?Guo-Qiang Lin,?Zhi-Tao He*.?Asymmetric Remote Leaving Group-Promoted Propargylic Substitution.?ACS Catal.?2025,?15,?10030–10038.
16.?Yu-Feng Liang,?Han-Zhe Miao, Xin Wang, Guo-Qiang Lin, Zhi-Tao He*.?Asymmetric?N-1,5-Addition and Cascade: Facile Route to Various?N-Heterocycles.?ACS Catal.?2025,?15,?10685–10693.
15.?Chao Ma,?Liang Chen,?Zhi-Tao He*.?Asymmetric Intramolecular?O-Hydroximation of Alkynes.?CCS Chem.?2025, 7,?1168–1176.
14.?Ye-Wei Chen, Yehao Qiu, Yang Liu, Guo-Qiang Lin, John F. Hartwig*, Zhi-Tao He*.?Intermolecular asymmetric functionalization of unstrained C(sp3)–C(sp3) bonds in allylic substitution reactions.?Nat. Synth.?2024,?3,?1011–1020.
13.?Yang Liu, Ye-Wei Chen, Yuan-Xiang Yang, John F. Hartwig*, Zhi-Tao He*.?Asymmetric Amination of Unstrained C(sp3)–C(sp3) Bonds.?J. Am. Chem. Soc.?2024,?146,?29857–29864.
12.?Bo-Yuan Xie, Zhi-Tao He*.?Chemodivergent Tandem Hydroalkylation and Hydroalkenoxylation of Conjugated Enynes.?ACS Catal.?2024,?14,?9742–9751.?
11.?Zi-Han Li, Jiang-Shan Ma, Han-Yu Lu, Guo-Qiang Lin, Zhi-Tao He*.?Asymmetric Multicomponent Propargylations via Carbon Dioxide Shuttling and Fixation.?ACS Catal.?2024,?14, 11646?11656.
10.?Xian-Xiao Chen,?Hao Luo,?Ye-Wei Chen, Yang Liu,?Zhi-Tao He*.?Enantioselective Palladium-Catalyzed Directed Migratory Allylation of Remote Dienes.?Angew. Chem. Int. Ed.?2023,?62,?e202307628.
9.?Ming-Qiao Tang, Zi-Jiang Yang,?Zhi-Tao He*.?Asymmetric Formal sp2-Hydrocarbonations of Dienes and Alkynes via Palladium Hydride Catalysis.?Nat. Commun.?2023,?14, 6303.
8.?Yu-Ze Sun,?Zi-Yang Ren,?Yuan-Xiang Yang, Yang Liu, Guo-Qiang Lin*,?Zhi-Tao He*.?Asymmetric Substitution by Alkynyl Copper Driven Dearomatization and Rearomatization.?Angew. Chem. Int. Ed.?2023,?62,?e202314517.
7.?Shao-Qian Yang, Ai-Jun Han, Yang Liu, Xin-Yuan Tang, Guo-Qiang Lin*, Zhi-Tao He*.?Catalytic Asymmetric Hydroalkoxylation and Formal Hydration and Hydroaminoxylation of Conjugated Dienes.?J. Am. Chem. Soc.?2023,?145,?3915–3925.
6.?Xin Wang, Han-Zhe Miao, Guo-Qiang Lin*, Zhi-Tao He*. Ligand-Dictated Regiodivergent Allylic Functionalizations via Palladium-Catalyzed Remote Substitution.?Angew. Chem. Int. Ed.?2023,?62,?e202301556.
5.?Jiang-Shan Ma,?Han-Yu Lu,?Ye-Wei Chen, Wei-Cheng Zhao, Yu-Ze Sun, Rui-Peng Li,?Hu-Xiao Wang, Guo-Qiang Lin*,?Zhi-Tao He*.?Copper-Catalyzed Convergent Regio- and Enantioselective?Alkynylallylic Substitution.?Nat. Synth.?2023,?2, 37–48.
4.?Yu-Chao Wang,?Zhao-Xin Xiao,?Miao Wang,?Shao-Qian Yang, Jin-Biao Liu, Zhi-Tao He*.?Umpolung Asymmetric 1,5-Conjugate Addition via Palladium Hydride Catalysis.?Angew. Chem. Int. Ed.?2023,?62,?e202215568.?
3.?Wei-Cheng Zhao,?Rui-Peng Li,?Chao Ma, Qi-Ying Liao, Miao Wang, Zhi-Tao He*. Stereoselective?gem-C,B-Glycosylation via 1,2-Boronate Migration.?J. Am. Chem. Soc.?2022,?144,?2460–2467.
2.?Ye-Wei Chen,?Yang Liu,?Han-Yu Lu,?Guo-Qiang Lin*, Zhi-Tao He*.?Palladium-Catalyzed Regio- and Enantioselective Migratory Allylic C(sp3)-H Functionalization.?Nat. Commun.?2021,?12,?5626.
1.?Shao-Qian Yang,?Yi-Fan Wang,?Wei-Cheng Zhao, Guo-Qiang Lin*, Zhi-Tao He*.?Stereodivergent Synthesis of Tertiary Fluoride-Tethered Allenes via Copper and Palladium Dual Catalysis.?J. Am. Chem. Soc.?2021,?143,?7285–7291.

